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GW 841819X
CAS No. 146135-18-4
GW 841819X ( GW841819X )
产品货号. M11985 CAS No. 146135-18-4
GW 841819X is an analogue of (+)-JQ1 and a novel inhibitor of BET bromodomain.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥7857 | 有现货 |
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| 50MG | ￥16038 | 有现货 |
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| 100MG | ￥20250 | 有现货 |
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| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称GW 841819X
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述GW 841819X is an analogue of (+)-JQ1 and a novel inhibitor of BET bromodomain.
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产品描述GW 841819X is an analogue of (+)-JQ1 and a novel inhibitor of BET bromodomain that displays activity in vivo against NUT-midline carcinoma, multiple myeloma, mixed-lineage leukemia, and acute myeloid leukemia.
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同义词GW841819X
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通路Chromatin/Epigenetic
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靶点Bromodomain
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受体Bromodomain
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研究领域——
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适应症——
化学信息
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CAS Number146135-18-4
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分子量487.94
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分子式C26H22ClN5O3
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纯度>98% (HPLC)
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溶解度——
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SMILESO=C(OCC1=CC=CC=C1)N[C@H]2C3=NN=C(C)N3C4=CC=C(OC)C=C4C(C5=CC=C(Cl)C=C5)=N2
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化学全称(R)-benzyl (6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-4-yl)carbamate
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Chung CW, et al. J Med Chem. 2011 Jun 9;54(11):3827-38.
2. Baud MG, et al. Science. 2014 Oct 31;346(6209):638-41.
2. Baud MG, et al. Science. 2014 Oct 31;346(6209):638-41.
产品手册
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